Cialis (Tadalafil) 5 mg – 30 Tablets
Description
Biochem Cialis (Tadalafil) 5 mg – 30 Tablets | Oral PDE5 Inhibitor
Biochem Cialis (Tadalafil) 5 mg – 30 Tablets is an oral pharmaceutical product. This product contains tadalafil, a selective phosphodiesterase type 5 (PDE5) inhibitor used in the medical management of erectile dysfunction and certain urinary symptoms associated with benign prostatic hyperplasia.
Tadalafil belongs to the PDE5 inhibitor class, which also includes sildenafil, vardenafil, and avanafil. These medications act through the nitric oxide–cyclic guanosine monophosphate (NO–cGMP) signaling pathway.
Tadalafil is associated with the pharmaceutical brand name Cialis. Its prolonged duration of pharmacological activity distinguishes it from several other medications in the same class.
Tadalafil selectively inhibits PDE5, an enzyme responsible for breaking down cyclic guanosine monophosphate (cGMP). By slowing cGMP degradation, tadalafil enhances nitric oxide-mediated smooth muscle relaxation.
In penile erectile tissue, this mechanism supports increased blood flow during sexual stimulation. Tadalafil does not independently produce an erection in the absence of appropriate sexual stimulation.
Tadalafil also influences smooth muscle signaling in tissues associated with the prostate, bladder, and lower urinary tract.
The compound has established medical applications for erectile dysfunction and, in certain jurisdictions, signs and symptoms of benign prostatic hyperplasia (BPH).
Tadalafil is also used in specialized pulmonary arterial hypertension treatment under distinct product indications and medical supervision.
The 5 mg strength is commonly associated with certain prescribed once-daily tadalafil regimens, but tablet strength alone does not determine the appropriate regimen for an individual patient.
Biochem Cialis 5 mg contains 5 mg of tadalafil per tablet, with 30 tablets per package. This provides 150 mg of tadalafil per package.
The Cialis brand name is associated with authorized tadalafil products. Its appearance in a Biochem description does not independently establish that Biochem tablets are authentic branded Cialis or an approved interchangeable generic.
| Specification | Details |
|---|---|
| Product Name | Biochem Cialis |
| Generic Name | Tadalafil |
| Active Ingredient | Tadalafil |
| Associated Brand | Cialis |
| Tablet Strength | 5 mg |
| Package Quantity | 30 Tablets |
| Total Active Ingredient | 150 mg |
| Dosage Form | Oral Tablets |
| Pharmacological Class | Phosphodiesterase Type 5 Inhibitor |
| Drug Abbreviation | PDE5 Inhibitor |
| Molecular Formula | C₂₂H₁₉N₃O₄ |
| Molecular Weight | Approximately 389.40 g/mol |
| Molecular Target | Phosphodiesterase Type 5 |
| Primary Pathway | Nitric Oxide–cGMP |
| Primary Mechanism | Inhibition of cGMP Breakdown |
| Primary Clinical Application | Erectile Dysfunction |
| Additional Clinical Application | Benign Prostatic Hyperplasia Symptoms |
| Other Tadalafil Indication | Pulmonary Arterial Hypertension Under Separate Product Indications |
| Sexual Stimulation Required for Erectile Effect | Yes |
| Approximate Elimination Half-Life | 17.5 Hours |
| Potential Erectile-Response Window | Up to Approximately 36 Hours |
| Primary Metabolic Enzyme | CYP3A4 |
| Metabolism | Predominantly Hepatic |
| Elimination | Mainly as Metabolites Through Feces and Urine |
| Administration Route | Oral |
| Food Effect | No Clinically Significant Effect on Overall Absorption |
| Nitrate Combination | Contraindicated |
| Riociguat Combination | Contraindicated |
| Prescription Classification | Prescription Medication in Many Jurisdictions |
| Excipients | Product-Specific Composition Not Confirmed |
| Manufacturing Specifications | Not Independently Verified |
1. Selectively Inhibits Phosphodiesterase Type 5
Tadalafil inhibits PDE5, an enzyme involved in regulating cGMP concentrations in smooth muscle cells.
PDE5 inhibition slows cGMP degradation and allows nitric oxide-mediated signaling to persist longer.
2. Supports Erectile Function Through Vascular Smooth Muscle Relaxation
During sexual stimulation, nitric oxide release increases cGMP production in penile tissue.
Tadalafil enhances this pathway by reducing cGMP breakdown, supporting smooth muscle relaxation and increased penile blood flow.
3. Has a Relatively Prolonged Duration of Action
Tadalafil has an elimination half-life of approximately 17.5 hours.
For erectile dysfunction, its effects may support responsiveness to sexual stimulation for up to approximately 36 hours after an appropriate dose. This does not mean an erection lasts for 36 hours.
4. Has Established Applications in Erectile Dysfunction
Tadalafil is used in selected patients with erectile dysfunction, a condition involving difficulty achieving or maintaining an erection sufficient for sexual activity.
The appropriate treatment depends on cardiovascular health, medications, underlying causes, and clinical assessment.
5. Has Established Applications in Benign Prostatic Hyperplasia
Tadalafil may improve certain lower urinary tract symptoms associated with BPH.
Its effects involve smooth muscle signaling and are not equivalent to directly shrinking prostate tissue.
6. Undergoes CYP3A4-Mediated Metabolism
Tadalafil is metabolized primarily by CYP3A4.
Strong CYP3A4 inhibitors or inducers may substantially alter tadalafil exposure. Kidney or liver impairment can also affect treatment decisions.
7. Requires Important Cardiovascular and Medication Safety Precautions
Tadalafil can lower blood pressure. It must not be combined with nitrates or riociguat because dangerous hypotension may occur.
Other important risks include headache, flushing, indigestion, back pain, muscle aches, dizziness, and rare sudden vision or hearing loss. An erection lasting more than four hours requires emergency medical attention.
Step 1 – Oral Administration and Absorption
Tadalafil is absorbed following oral administration and enters systemic circulation.
Step 2 – Distribution to PDE5-Expressing Tissues
Tadalafil reaches tissues containing PDE5, including vascular and urogenital smooth muscle.
Step 3 – Inhibition of cGMP Degradation
Tadalafil inhibits PDE5 and slows the breakdown of cGMP.
Step 4 – Enhancement of Nitric Oxide-Mediated Relaxation
During sexual stimulation, enhanced cGMP signaling supports smooth muscle relaxation and penile blood flow.
Step 5 – Metabolism and Elimination
Tadalafil undergoes hepatic metabolism, primarily through CYP3A4. Its metabolites are eliminated through fecal and urinary pathways.
The Biochem Cialis 5 mg presentation includes these characteristics:
- Tadalafil as the active ingredient.
- 5 mg per tablet.
- 30 tablets per package.
- 150 mg total tadalafil content.
- Oral tablet formulation.
- PDE5 inhibitor classification.
- Nitric oxide–cGMP pathway activity.
- Smooth muscle relaxation mechanism.
- Established erectile dysfunction indication.
- Established BPH symptom indication.
- Approximately 17.5-hour elimination half-life.
- Potential erectile-response window up to approximately 36 hours.
- Sexual stimulation required for erectile response.
- Primarily CYP3A4-mediated metabolism.
- Important cardiovascular safety considerations.
- Contraindication with nitrate medications.
- Contraindication with riociguat.
- Potential interactions with alpha-blockers and other blood-pressure-lowering medicines.
- Product-specific excipients requiring confirmation.
- Identity and content uniformity requiring analytical verification.
The precise excipients, manufacturing specifications, and independent quality testing of Biochem Cialis 5 mg have not been verified.
United States
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Canada
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United Kingdom
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Germany
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France
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Spain
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Italy
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Portugal
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Netherlands
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Belgium
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Switzerland
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Austria
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Sweden
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Norway
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Denmark
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Finland
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Poland
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Czech Republic
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Romania
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Greece
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Ireland
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Colombia
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Argentina
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México
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Perú
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Venezuela
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Ecuador
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Biochem Cialis (Tadalafil) 5mg | 30 Tablets | PDE5 Inhibitor
Learn about Biochem Cialis 5mg, 30 tablets. This product contains tadalafil, a PDE5 inhibitor used in selected erectile dysfunction and benign prostatic hyperplasia treatment settings.
Biochem Cialis (Tadalafilo) 5mg | 30 Tabletas | Inhibidor PDE5
Conoce Biochem Cialis 5mg, 30 tabletas. Este producto contiene tadalafilo, un inhibidor PDE5 utilizado en determinados tratamientos de la disfunción eréctil y los síntomas de hiperplasia prostática benigna.
biochem-cialis-tadalafil-5mg-30-tablets
biochem-cialis-tadalafilo-5mg-30-tabletas
Biochem Cialis Tadalafil 5mg, 30 oral tablets containing tadalafil, a phosphodiesterase type 5 inhibitor associated with nitric oxide–cGMP signaling and smooth muscle relaxation.
Biochem Cialis Tadalafilo 5mg, 30 tabletas orales que contienen tadalafilo, un inhibidor de la fosfodiesterasa tipo 5 relacionado con la señalización del óxido nítrico y GMPc.